Entry | Reagent | Additive | Base | Yield [%] b |
---|
1 | DMTMM | - | NMM | 89 |
2 | WSCI | HONB | DIEA | 25 |
3 | WSCI | HOSu | DIEA | 32 |
4 | WSCI | Sulfo-HOSu | DIEA | 71 |
- a Reactions were carried out between H-Leu-NH2 and water-dispersible Boc-Phe-OH nanoparticles. b The yield of peptides was calculated from analytical HPLC profiles.